产品详情

Paliperidone Palmitate,50MG,SML4082-50MG,Sigma

销售价: ¥ 3064.50 / 件
优    惠: 请询价
订货号 0BP8262
品牌型号 SML4082-50MG
货期 询货期
最小订货量 1件
产品介绍 Product Description

Biochem/physiol Actions

Prodrug form of paliperidone, is a long-acting injectable antipsychotic that targets dopamine and serotonin receptors.


Paliperidone palmitate is a long-acting injectable form of paliperidone, an atypical antipsychotic that targets dopamine D2 and serotonin 5-HT2A receptors to alleviate schizophrenia symptoms through neurotransmission regulation. Paliperidone palmitate also interacts with α1/α2 adrenergic and H1 histaminergic receptors, influencing both its therapeutic effects and side effect profile. The formulation′s sustained release mechanism promotes gradual absorption, ensuring stable drug levels for prolonged efficacy.


技术参数 Specifications
Quality Segment100
assay≥98% (HPLC)
formpowder
color white to beige
solubilitysoluble (DMSO:TFA, 2 mg/mL, clear (add 1 drop TFA))
storage temp.-10 to -25°C
SMILES stringFc1cc2[o]nc(c2cc1)C3CCN(CC3)CCC4=C(NC5=C(CCCN5C4=O)OC(=O)CCCCCCCCCCCCCCC)C
InChI keyYOSKWMGLLZWACB-UHFFFAOYSA-N
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