产品介绍
Product Description
Biochem/physiol Actions
Neutral antagonist of the μ-opioid receptor. A reduction of withdrawal effects associated with neutral μ-opioid receptor antagonists may offer advantages in treating opioid overdose and addiction.
Features and Benefits
This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
技术参数
Specifications
| Quality Level | 100 |
| assay | ≥96% (HPLC) |
| form | powder |
| drug control | regulated under CDSA - not available from Sigma-Aldrich Canada |
| color | white |
| solubility | DMSO: ~12 mg/mL,H2O: insoluble |
| storage temp. | 2-8°C |
| SMILES string | [H]O[H].O[C@@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5O[C@@H]1[C@]2(CCN3CC6CC6)c45 |
| InChI | 1S/C20H25NO4.H2O/c22-13-4-3-12-9-15-20(24)6-5-14(23)18-19(20,16(12)17(13)25-18)7-8-21(15)10-11-1-2-11;/h3-4,11,14-15,18,22-24H,1-2,5-10H2;1H2/t14-,15-,18+,19+,20-;/m1./s1 |
| InChI key | VHGGWFVHXKTOPK-CDHBEYIESA-N |
