产品介绍
Product Description
Biochem/physiol Actions
Orally bioavailable, potent, and selective partial agonist of serotonin 5-HT1A receptor; non-sedative anxiolytic and antidepressant drug.
Gepirone hydrochloride is an orally bioavailable, non-sedative anxiolytic and antidepressant drug of the buspirone family with a unique mechanism of action that differs from other antidepressants and anxiolytic drugs. Gepirone acts as a partial serotonin 5-HT1A receptor agonist with differential action at pre-and postsynaptic 5-HT1A receptors. Gepirone is much more efficacious than selective serotonin reuptake inhibitors (SSRIs) without causing sexual dysfunction.
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Hygroscopic
技术参数
Specifications
| Quality Level | 100 |
| assay | ≥98% (HPLC) |
| form | powder |
| storage condition | desiccated |
| color | white to beige |
| solubility | H2O: 2 mg/mL, clear |
| storage temp. | -10 to -25°C |
| SMILES string | O=C1N(C(CC(C1)(C)C)=O)CCCCN2CCN(C3=NC=CC=N3)CC2.[xHCl] |
