产品介绍
Product Description
Biochem/physiol Actions
CBP/p300 Bromodomain inhibitor
CPI-637 is a cell penetrant, selective and potent CBP/p300 bromodomain inhibitor.
技术参数
Specifications
| assay | ≥98% (HPLC) |
| form | powder |
| optical activity | [α]/D -39 to -49°, c = 1.0 in chloroform-d |
| color | white to beige |
| solubility | DMSO: 2 mg/mL, clear |
| storage temp. | −20°C |
| SMILES string | [n]1(ncc(c1)c2n[n](c3c2cc(cc3)c4c5c(ccc4)NC(=O)C[C@H](N5)C)C)C |
| InChI | 1S/C22H22N6O/c1-13-9-20(29)25-18-6-4-5-16(22(18)24-13)14-7-8-19-17(10-14)21(26-28(19)3)15-11-23-27(2)12-15/h4-8,10-13,24H,9H2,1-3H3,(H,25,29)/t13-/m1/s1 |
| InChI key | BFTKDWYIRJGJCA-CYBMUJFWSA-N |
